Receptors database
Experimental GPCR structures studied in GPCR-IFP.
Protein | Specie | PDB code | Ligand type | More |
cxcr4 | human | 3OE6, 3OE9, 3ODU, 3OE8, 3OE0, 4RWS | antagonist | |
opsd | todpa | 3AYN, 2Z73 | inverse agonist | |
opsd | bovin | 3C9L, 1L9H, 3OAX, 3C9M, 2PED, 1F88, 2J4Y, 1HZX, 1U19, 1GZM | inverse agonist | |
opsd | todpa | 3AYM, 4WW3 | agonist | |
ox1r | human | 6TQ4, 6TP3, 6V9S, 6TP4, 4ZJC, 6TQ9, 6TOT, 6TQ6, 6TQ7, 4ZJ8, 6TOD, 6TOS, 6TP6, 6TO7 | antagonist | |
ada2b | human | 6K41 | agonist | |
s1pr3 | human | 7EW3, 7EW2, 7C4S, 7EW4 | agonist | |
aa2ar | human | 2YDV, 4UG2, 5G53, 4UHR, 2YDO, 5WF6, 5WF5, 3QAK | agonist | |
adrb1 | melga | 4BVN, 3ZPR, 2YCW, 2VT4, 2YCY, 5F8U, 3ZPQ, 2YCX | antagonist | |
aa2ar | human | 5IUA, 5UVI, 5VRA, 3UZA, 6LPK, 4EIY, 5NM4, 5OLG, 5UIG, 5N2R, 6LPJ, 5IU8, 5OLV, 3EML, 3VGA, 3PWH, 5K2A, 6ZDR, 5OLH, 7RM5, 6ZDV, 5OLZ, 5MZP, 5OM4, 6WQA, 5K2B, 3REY, 6LPL, 3VG9, 5OM1, 5K2C, 5NM2, 6PS7, 5IUB, 6AQF, 5MZJ, 6GT3, 5IU7, 3UZC, 5JTB, 5IU4, 6JZH, 5K2D, 5OLO, 5NLX, 6S0L, 6S0Q | antagonist | |
oprd | human | 4RWD, 4N6H, 4RWA | antagonist | |
5ht1b | human | 6G79, 4IAR, 4IAQ | agonist | |
adrb2 | human | 3D4S, 5JQH, 3NY8, 3NY9, 2RH1, 5D5A, 5D6L | inverse agonist | |
adrb1 | melga | 2Y03, 2Y02, 4AMI, 6H7L, 6H7N, 6H7O, 6TKO, 7JJO, 6H7M, 6IBL, 6H7J | agonist | |
adrb2 | human | 7DHR, 4QKX, 4LDL, 3PDS, 7DHI, 6NI3, 4LDO, 4LDE, 7BZ2, 6MXT, 3P0G, 3SN6 | agonist | |
5ht2a | human | 6WH4 | inverse agonist | |
cltr1 | human | 6RZ5, 6RZ4 | antagonist | |
ffar1 | human | 4PHU, 5TZR | agonist | |
opsd | bovin | 5DYS, 6FK8, 6OYA, 6FK7, 2G87, 2HPY, 3PXO, 4A4M, 6FK6, 6FKB, 3PQR, 5EN0, 6OY9, 6FKC, 2X72, 6FUF, 6FKD, 6FK9, 6FKA | agonist | |
5ht2b | human | 4IB4, 5TUD, 5TVN, 6DRY, 4NC3 | agonist | |
adrb1 | human | 7BVQ | inverse agonist | |
ednrb | human | 6K1Q | inverse agonist | |
aa2ar | human | 7ARO | agonist (partial) | |
5ht2c | human | 6BQG | agonist | |
5ht2a | human | 6WHA, 6WGT | agonist | |
acm2 | human | 5ZK3, 5ZKC, 5YC8, 3UON, 5ZK8, 5ZKB | antagonist | |
cckar | human | 7F8U, 7F8Y | antagonist | |
s1pr1 | human | 3V2Y, 3V2W | antagonist | |
acm3 | rat | 4U15, 5ZHP, 4DAJ | antagonist | |
agtr1 | human | 4ZUD | inverse agonist | |
pe2r4 | human | 7D7M | agonist | |
nk1r | human | 6HLO, 6HLL, 6J21, 6E59, 6HLP, 6J20 | antagonist | |
ednrb | human | 5X93 | antagonist | |
par1 | human | 3VW7 | antagonist | |
mtr1a | human | 7DB6, 6ME3, 6ME5, 6ME4, 6PS8, 6ME2 | agonist | |
npy2r | human | 7DDZ | antagonist | |
acm1 | human | 6ZFZ, 6ZG4, 6ZG9, 6OIJ | agonist | |
oprx | human | 5DHG, 5DHH, 4EA3 | antagonist | |
aa1r | human | 5UEN | antagonist | |
sucr1 | rat | 6RNK, 6Z10 | antagonist | |
agtr2 | human | 5UNG, 5UNH, 5UNF | antagonist | |
ada2a | human | 6KUX | antagonist | |
s1pr5 | human | 7EW1 | agonist | |
oprd | human | 6PT2, 6PT3 | agonist | |
ptafr | human | 5ZKQ | inverse agonist | |
drd3 | human | 3PBL | antagonist | |
ox2r | human | 7L1V, 7L1U | agonist | |
5ht2c | human | 6BQH | inverse agonist | |
mc4r | human | 7F54, 7F55, 7F58, 7F53, 7AUE, 7PIU, 7PIV | agonist | |
oprk | human | 4DJH, 6VI4 | antagonist | |
5ht1e | human | 7E33 | agonist | |
pe2r3 | human | 6AK3, 6M9T | agonist | |
gnrhr | human | 7BR3 | antagonist | |
drd2 | human | 7JVR, 6VMS | agonist | |
oprk | human | 6B73 | agonist | |
cnr2 | human | 6PT0, 6KPF, 6KPC | agonist | |
drd3 | human | 7CMV, 7CMU | agonist | |
cltr2 | human | 6RZ6, 6RZ7, 6RZ9, 6RZ8 | antagonist | |
pe2r4 | human | 5YWY | antagonist | |
cnr2 | human | 5ZTY | antagonist | |
lpar1 | human | 4Z35, 4Z34, 4Z36 | antagonist | |
hrh1 | human | 3RZE | antagonist | |
lt4r1 | human | 7K15 | antagonist | |
drd4 | human | 5WIU, 5WIV | antagonist | |
5ht2a | human | 6A94, 6A93 | antagonist | |
cnr1 | human | 5U09 | inverse agonist | |
npy1r | human | 5ZBQ, 5ZBH | antagonist | |
5ht1f | human | 7EXD | agonist | |
ox2r | human | 5WS3, 6TPJ, 6TPG, 6TPN, 4S0V, 5WQC | antagonist | |
ccr5 | human | 4MBS, 6AKX, 6MEO, 5UIW, 6AKY | antagonist | |
ccr2 | human | 6GPS, 6GPX | antagonist | |
drd2 | human | 6CM4 | inverse agonist | |
gpbar | human | 7CFM | agonist | |
pd2r2 | human | 6D26, 7M8W, 6D27 | antagonist | |
ta2r | human | 6IIU, 6IIV | antagonist | |
p2y12 | human | 4PXZ | agonist | |
cnr1 | human | 5XR8, 6N4B, 5XRA, 6KPG, 7V3Z | agonist | |
adrb1 | melga | 4AMJ, 5A8E | inverse agonist | |
acm4 | human | 5DSG | antagonist | |
adrb1 | melga | 2Y00, 2Y01, 2Y04 | agonist (partial) | |
adrb2 | human | 3NYA, 6PS5, 6PS3, 6PS0, 6PS2, 6PS1, 6PS4, 6PRZ, 6PS6 | antagonist | |
oxyr | human | 6TPK | antagonist | |
mtr1b | human | 6ME8, 6ME6, 6ME9, 6ME7 | agonist | |
5ht2b | human | 6DRZ, 6DRX, 6DS0 | antagonist | |
acm2 | human | 4MQS | agonist | |
ghsr | human | 7F9Z, 7F9Y, 7NA7, 7NA8 | agonist | |
p2y12 | human | 4PY0 | agonist (partial) | |
ptafr | human | 5ZKP | antagonist | |
acm1 | human | 5CXV | antagonist | |
p2ry1 | human | 4XNW | antagonist | |
agtr1 | human | 4YAY | antagonist | |
adrb1 | human | 7BTS, 7BU7, 7BU6 | agonist | |
oprd | mouse | 4EJ4 | antagonist | |
ada2a | human | 6KUY | agonist (partial) | |
drd2 | human | 7DFP, 6LUQ | antagonist | |
c5ar1 | human | 5O9H | antagonist | |
ednrb | human | 6IGL | agonist (partial) | |
adrb3 | canlf | 7DH5 | agonist | |
drd4 | mouse | 6IQL | antagonist | |
drd1 | human | 7JVQ, 7JVP, 7CKW, 7CRH, 7JV5, 7CKX, 7CKY | agonist | |
gpr52 | human | 6LI0 | agonist | |
ada2c | human | 6KUW | antagonist | |
cnr1 | human | 5TGZ | antagonist | |
par2 | human | 5NDD | antagonist | |
ghsr | human | 6KO5 | antagonist | |
p2y12 | human | 4NTJ | antagonist | |
5ht1b | human | 7C61 | antagonist | |
pe2r2 | human | 7CX2, 7CX4, 7CX3 | agonist | |
5ht1a | human | 7E2Y | agonist | |
5ht1d | human | 7E32 | agonist | |
hrh1 | human | 7DFL | agonist | |
5ht1a | human | 7E2Z | agonist (partial) | |
gp139 | human | 7VUJ, 7VUG, 7VUI, 7VUH | agonist | |
mrgx2 | human | 7VV6, 7VV0, 7S8O, 7VDH, 7S8N, 7VV3, 7VDM, 7VUZ, 7VV5, 7VDL, 7S8L, 7VV4, 7VUY, 7S8M | agonist | |
s1pr1 | human | 7EO4, 7EO2, 7WF7 | agonist | |
5ht2a | human | 7VOE, 7VOD | agonist (partial) | |
mrgx4 | human | 7S8P | agonist |