Receptors database

Experimental GPCR structures studied in GPCR-IFP.


Protein Specie PDB code Ligand type More
human 3OE6, 3OE9, 3ODU, 3OE8, 3OE0, 4RWS antagonist
todpa 3AYN, 2Z73 inverse agonist
bovin 3C9L, 1L9H, 3OAX, 3C9M, 2PED, 1F88, 2J4Y, 1HZX, 1U19, 1GZM inverse agonist
todpa 3AYM, 4WW3 agonist
human 6TQ4, 6TP3, 6V9S, 6TP4, 4ZJC, 6TQ9, 6TOT, 6TQ6, 6TQ7, 4ZJ8, 6TOD, 6TOS, 6TP6, 6TO7 antagonist
human 6K41 agonist
human 7EW3, 7EW2, 7C4S, 7EW4 agonist
human 2YDV, 4UG2, 5G53, 4UHR, 2YDO, 5WF6, 5WF5, 3QAK agonist
melga 4BVN, 3ZPR, 2YCW, 2VT4, 2YCY, 5F8U, 3ZPQ, 2YCX antagonist
human 5IUA, 5UVI, 5VRA, 3UZA, 6LPK, 4EIY, 5NM4, 5OLG, 5UIG, 5N2R, 6LPJ, 5IU8, 5OLV, 3EML, 3VGA, 3PWH, 5K2A, 6ZDR, 5OLH, 7RM5, 6ZDV, 5OLZ, 5MZP, 5OM4, 6WQA, 5K2B, 3REY, 6LPL, 3VG9, 5OM1, 5K2C, 5NM2, 6PS7, 5IUB, 6AQF, 5MZJ, 6GT3, 5IU7, 3UZC, 5JTB, 5IU4, 6JZH, 5K2D, 5OLO, 5NLX, 6S0L, 6S0Q antagonist
human 4RWD, 4N6H, 4RWA antagonist
human 6G79, 4IAR, 4IAQ agonist
human 3D4S, 5JQH, 3NY8, 3NY9, 2RH1, 5D5A, 5D6L inverse agonist
melga 2Y03, 2Y02, 4AMI, 6H7L, 6H7N, 6H7O, 6TKO, 7JJO, 6H7M, 6IBL, 6H7J agonist
human 7DHR, 4QKX, 4LDL, 3PDS, 7DHI, 6NI3, 4LDO, 4LDE, 7BZ2, 6MXT, 3P0G, 3SN6 agonist
human 6WH4 inverse agonist
human 6RZ5, 6RZ4 antagonist
human 4PHU, 5TZR agonist
bovin 5DYS, 6FK8, 6OYA, 6FK7, 2G87, 2HPY, 3PXO, 4A4M, 6FK6, 6FKB, 3PQR, 5EN0, 6OY9, 6FKC, 2X72, 6FUF, 6FKD, 6FK9, 6FKA agonist
human 4IB4, 5TUD, 5TVN, 6DRY, 4NC3 agonist
human 7BVQ inverse agonist
human 6K1Q inverse agonist
human 7ARO agonist (partial)
human 6BQG agonist
human 6WHA, 6WGT agonist
human 5ZK3, 5ZKC, 5YC8, 3UON, 5ZK8, 5ZKB antagonist
human 7F8U, 7F8Y antagonist
human 3V2Y, 3V2W antagonist
rat 4U15, 5ZHP, 4DAJ antagonist
human 4ZUD inverse agonist
human 7D7M agonist
human 6HLO, 6HLL, 6J21, 6E59, 6HLP, 6J20 antagonist
human 5X93 antagonist
human 3VW7 antagonist
human 7DB6, 6ME3, 6ME5, 6ME4, 6PS8, 6ME2 agonist
human 7DDZ antagonist
human 6ZFZ, 6ZG4, 6ZG9, 6OIJ agonist
human 5DHG, 5DHH, 4EA3 antagonist
human 5UEN antagonist
rat 6RNK, 6Z10 antagonist
human 5UNG, 5UNH, 5UNF antagonist
human 6KUX antagonist
human 7EW1 agonist
human 6PT2, 6PT3 agonist
human 5ZKQ inverse agonist
human 3PBL antagonist
human 7L1V, 7L1U agonist
human 6BQH inverse agonist
human 7F54, 7F55, 7F58, 7F53, 7AUE, 7PIU, 7PIV agonist
human 4DJH, 6VI4 antagonist
human 7E33 agonist
human 6AK3, 6M9T agonist
human 7BR3 antagonist
human 7JVR, 6VMS agonist
human 6B73 agonist
human 6PT0, 6KPF, 6KPC agonist
human 7CMV, 7CMU agonist
human 6RZ6, 6RZ7, 6RZ9, 6RZ8 antagonist
human 5YWY antagonist
human 5ZTY antagonist
human 4Z35, 4Z34, 4Z36 antagonist
human 3RZE antagonist
human 7K15 antagonist
human 5WIU, 5WIV antagonist
human 6A94, 6A93 antagonist
human 5U09 inverse agonist
human 5ZBQ, 5ZBH antagonist
human 7EXD agonist
human 5WS3, 6TPJ, 6TPG, 6TPN, 4S0V, 5WQC antagonist
human 4MBS, 6AKX, 6MEO, 5UIW, 6AKY antagonist
human 6GPS, 6GPX antagonist
human 6CM4 inverse agonist
human 7CFM agonist
human 6D26, 7M8W, 6D27 antagonist
human 6IIU, 6IIV antagonist
human 4PXZ agonist
human 5XR8, 6N4B, 5XRA, 6KPG, 7V3Z agonist
melga 4AMJ, 5A8E inverse agonist
human 5DSG antagonist
melga 2Y00, 2Y01, 2Y04 agonist (partial)
human 3NYA, 6PS5, 6PS3, 6PS0, 6PS2, 6PS1, 6PS4, 6PRZ, 6PS6 antagonist
human 6TPK antagonist
human 6ME8, 6ME6, 6ME9, 6ME7 agonist
human 6DRZ, 6DRX, 6DS0 antagonist
human 4MQS agonist
human 7F9Z, 7F9Y, 7NA7, 7NA8 agonist
human 4PY0 agonist (partial)
human 5ZKP antagonist
human 5CXV antagonist
human 4XNW antagonist
human 4YAY antagonist
human 7BTS, 7BU7, 7BU6 agonist
mouse 4EJ4 antagonist
human 6KUY agonist (partial)
human 7DFP, 6LUQ antagonist
human 5O9H antagonist
human 6IGL agonist (partial)
canlf 7DH5 agonist
mouse 6IQL antagonist
human 7JVQ, 7JVP, 7CKW, 7CRH, 7JV5, 7CKX, 7CKY agonist
human 6LI0 agonist
human 6KUW antagonist
human 5TGZ antagonist
human 5NDD antagonist
human 6KO5 antagonist
human 4NTJ antagonist
human 7C61 antagonist
human 7CX2, 7CX4, 7CX3 agonist
human 7E2Y agonist
human 7E32 agonist
human 7DFL agonist
human 7E2Z agonist (partial)
human 7VUJ, 7VUG, 7VUI, 7VUH agonist
human 7VV6, 7VV0, 7S8O, 7VDH, 7S8N, 7VV3, 7VDM, 7VUZ, 7VV5, 7VDL, 7S8L, 7VV4, 7VUY, 7S8M agonist
human 7EO4, 7EO2, 7WF7 agonist
human 7VOE, 7VOD agonist (partial)
human 7S8P agonist